Elacytarabine

名字：Elacytarabine
描述：Description: Elacytarabine, also known as CP-4055, is the lipophilic 5'-elaidic acid ester of the deoxycytidine analog cytosine arabinoside (cytarabine; Ara-C) with potential antineoplastic activity. As a prodrug, CP-4055 is converted intracellularly into cytarabine triphosphate by deoxycytidine kinase and subsequently competes with cytidine for incorporation into DNA, thereby inhibiting DNA synthesis. Compared to cytarabine, CP-4055 shows increased cellular uptake and retention, resulting in increased activation by deoxycytidine kinase to cytarabine triphosphate, decreased deamination and deactivation by deoxycytidine deaminase, and increased inhibition of DNA synthesis. This agent also inhibits RNA synthesis, an effect not seen with cytarabine.
规格:10mg;100mg;1g;25mg;200mg;2g;50mg;500mg;5g;
理论分析：THEORETICAL ANALYSIS
MedKoo Cat#: 201195
Name: Elacytarabine
CAS#: 188181-42-2
Chemical Formula: C27H45N3O6
Exact Mass: 507.33084
Molecular Weight: 507.6627
Elemental Analysis: C, 63.88; H, 8.93; N, 8.28; O, 18.91
技术数据：Appearance: Solid powder Purity: >98% (or refer to the Certificate of Analysis) Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs. Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years). Solubility: Soluble in DMSO, not in water Shelf Life: >2 years if stored properly Drug Formulation: This drug may be formulated in DMSO Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months). Harmonized System Code: 293490

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