名字：Fimasartan featured描述：Description: Fimasartan is a non-peptide angiotensin II receptor antagonist (ARB) used for the treatment of hypertension and heart failure. Through oral administration, fimasartan blocks angiotensin II receptor type 1 (AT1 receptors), reducing pro-hypertensive actions of ang...
名字：Fulvestrant featured描述：Description: Fulvestrant is a synthetic estrogen receptor antagonist. Unlike tamoxifen (which has partial agonist effects) and the aromatase inhibitors (which reduce the estrogen available to tumor cells), fulvestrant binds competitively to estrogen receptors in breast canc...
名字：GNE-495 new featured描述：Description: GNE-495 is a potent and selective MAP4K4 Inhibitor with efficacy in retinal angiogenesis. GNE-495 showed excellent potency and good PK and was used to demonstrate in vivo efficacy in a retinal angiogenesis model recapitulating effects that were observed in the ...
名字：GSK-F1描述：Description: GSK-F1 is a novel potent inhibitor of PI4KA.规格:理论分析：THEORETICAL ANALYSISMedKoo Cat#: 527468Name: GSK-F1CAS#: 1402345-92-9Chemical Formula: C27H18F5N5O4SExact Mass: 603.1Molecular Weight: 603.524Elemental Analysis: C, 53.73; H, 3.01; F, 15.74; N, 11.60; O, 10.60; S, 5.31技术数据：...
名字：HTS01037 featured描述：Description: HTS01037 is an inhibitor of fatty acid binding proteins (FABPs), which acts as an antagonist of protein-protein interactions mediated by FABPs, in particular adipocyte FABP.规格:5mg;10mg;25mg;理论分析：THEORETICAL ANALYSISMedKoo Cat#: 531956Name: HTS01037CAS#: 682741-29-...
名字：INI-43描述：Description: INI-43 is a novel Inhibitor of Nuclear Import-43, showing a significant cytotoxic effect on various cervical and oesophageal cancer cell lines by targeting Kpnß1.规格:理论分析：THEORETICAL ANALYSISMedKoo Cat#: 527034Name: INI-43CAS#: 881046-01-1Chemical Formula: C22H23N7Exact Mass:...
名字：JNJ-5207852 featured描述：Description: JNJ-5207852 is a potent and selective H3 antagonist with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor. JNJ-5207852 is selective for the H3 receptor, with negligible binding to other receptors, transporters and ion channels at 1 microm. JN...
名字：L-2286描述：Description: L-2286 is a novel PARP inhibitor. L-2286 exerted significant protective effect against ischemia-reperfusion-induced myocardial injury in both experimental models. More importantly, L-2286 facilitated the ischemia-reperfusion-induced activation of Akt, extracellular signal-re...
名字：LGD-3303 new featured描述：Description: LGD-3303 is a drug which acts as a selective androgen receptor modulator (SARM), with good oral bioavailability. It is a selective agonist for the androgen receptor, producing functional selectivity with effective dissociation of anabolic and androgenic effect...
名字：LY 207702描述：Description: LY 207702 is a difluorinated purine nucleoside that exhibits antitumor activity in preclinical models.规格:理论分析：THEORETICAL ANALYSISMedKoo Cat#: 525511Name: LY 207702CAS#: 103828-81-5Chemical Formula: C10H12F2N6O3Exact Mass: 302.0939Molecular Weight: 302.24Elemental Analysi...
