名字：UK 357903描述：Description: UK 357903 is a phosphodiesterase 5A (PDE5A) inhibitor potentially for the treatment of erectile dysfunction.规格:理论分析：THEORETICAL ANALYSISMedKoo Cat#: 529215Name: UK 357903CAS#: 247580-98-9Chemical Formula: C27H34N8O5SExact Mass: 582.2373Molecular Weight: 582.68Elemental An...
名字：Voglibose featured描述：Description: Voglibose is an alpha-glucosidase inhibitor used for lowering post-prandial blood glucose levels in people with diabetes mellitus. Voglibose delays the absorption of glucose thereby reducing the risk of macrovascular complications. Voglibose was first launched in...
名字：XK469描述：Description: XK489 is a synthetic quinoxaline phenoxypropionic acid derivative with proapoptotic and antiproliferative activities. R(+)XK469 selectively inhibits topoisomerase II-beta, blocks activation of MEK/MAPK signaling kinases, stimulates caspases, and upregulates p53-dependent prot...
名字：ZM 230487描述：Description: ZM 230487 is a 5-lipoxygenase inhibitor.规格:理论分析：THEORETICAL ANALYSISMedKoo Cat#: 526584Name: ZM 230487CAS#: 155944-23-3Chemical Formula: C24H26FNOExact Mass: 411.1846Molecular Weight: 411.4734Elemental Analysis: C, 70.06; H, 6.37; F, 4.62; N, 3.40; O, 15.55技术数据：Appearance...
名字：SLM6描述：Description: SLM6 is an inhibitor of cyclin-dependent kinase-9 (CDK9). It exhibits potent anti-multiple myeloma activity.规格:理论分析：THEORETICAL ANALYSISMedKoo Cat#: 561772Name: SLM6CAS#: 22242-91-7Chemical Formula: C12H17N7O4Exact Mass: 323.1342Molecular Weight: 323.31Elemental Analysis: C, 4...
名字：STF-62247 featured描述：Description: STF-62247 shows selective toxicity and growth inhibition of renal cells lacking VHL; 25-fold greater sensitivity observed for cells with VHL deficiency compared to wild-type (VHL+).规格:10mg;25mg;理论分析：THEORETICAL ANALYSISMedKoo Cat#: 531307Name: STF-62247CAS#: 3157...
名字：Talniflumate featured描述：Description: Talniflumate is a novel potent and selective inhibitor of core mucin-synthesizing enzyme GCNT3 (core 2b-1,6 N-acetylglucosaminyltrans-ferase).规格:200mg;500mg;1g;理论分析：THEORETICAL ANALYSISMedKoo Cat#: 526070Name: TalniflumateCAS#: 66898-62-2Chemical Formula: C21H...
名字：TG100435描述：Description: TG100435 is a potent, orally active Src inhibitor with desirable PK properties, demonstrated activity in human tumor cell lines and in animal models of tumor growth.规格:理论分析：THEORETICAL ANALYSISMedKoo Cat#: 406147Name: TG100435CAS#: NONEChemical Formula: C26H25Cl2N5OExact M...
名字：TPOP146描述：Description: TPOP146 is a potent and selective CBP/P300 Benzoxazepine Bromodomain Inhibitor. TPOP146 showed 134 nM affinity for CBP with excellent selectivity over other bromodomains. Deregulation of CBP/P300 has been reported in cancer and chromosomal rearrangement of the CBP/P300 locu...
名字：UK-371804 new featured描述：Description: UK-371804 is a potent and selective uPA inhibitor with excellent enzyme potency (Ki 10 nM) and selectivity profile (4000-fold versus tPA and 2700-fold versus plasmin). In vitro, UK-371804 is able to inhibit exogenous uPA in human chronic wound fluid (IC50=0.8...
